SCHEMBL3685873

SCHEMBL3685873

COc1ccccc1-c1ccc(C(=O)/C=C/c2ccccc2CN(C)C(C)(C)C)c(N2CCN(C)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HIF1A Q16665 1/20 0.40
KEAP1 Q14145 3/20 0.38
NFE2L2 Q16236 3/20 0.38
ABL1 P00519 1/20 0.38
HDAC3 O15379 2/20 0.38
HDAC4 P56524 2/20 0.38
HDAC1 Q13547 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686127 1.00 PTPN1 (0.41) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3686258 0.93 PTPN1 (0.43) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3685244 0.93 PTPN1 (0.43) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3685874 0.90 ALDH1A1 (0.41) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3695006 0.90 PTPN1 (0.44) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3691194 0.90 PTPN1 (0.41) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3693463 0.90 PTPN1 (0.44) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3684550 0.90 PTPN1 (0.41) PTPN1KDM4EMEN1ALDH1A1LMNA
SCHEMBL3693651 0.87 DRD2 (0.51) PTPN1KEAP1NFE2L2HDAC3HDAC4
SCHEMBL3683969 0.87 DRD2 (0.51) PTPN1KEAP1NFE2L2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed