SCHEMBL3695079

SCHEMBL3695079

CC(Cc1cccc(NC(=O)C(c2ccc(CN3N=C(c4ccccc4)OCC3=O)cc2)C2CCC(F)(F)C2)c1)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.37
PTGS2 P35354 9/20 0.36
MAOB P27338 2/20 0.35
ACKR3 P25106 4/20 0.34
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
C3AR1 Q16581 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL1080950 0.91 PTGES (0.38) PTGESMAOBACKR3C3AR1CHRM2
SCHEMBL1178170 0.90 PTGES (0.48) PTGESPTGS2MAOBC3AR1
SCHEMBL1080947 0.90 PTGES (0.38) PTGESMAOBACKR3C3AR1CHRM2
SCHEMBL1178056 0.89 PTGES (0.42) PTGESMAOBACKR3ITGB3ITGA2B
SCHEMBL1178655 0.86 PTGES (0.34) PTGESMAOBACKR3C3AR1CHRM2
SCHEMBL1178336 0.84 MAOB (0.34) MAOBC3AR1CHRM2CHRM1CHRM3
SCHEMBL1079856 0.82 PTGES (0.45) PTGESPTGS2MAOBACKR3
SCHEMBL3693615 0.82 ITGB3 (0.36) MAOBACKR3ITGB3ITGA2B
SCHEMBL1178131 0.81 PTGES (0.42) PTGESPTGS2MAOB
SCHEMBL1178561 0.81 PTGES (0.46) PTGESPTGS2MAOBACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed