SCHEMBL3695219

SCHEMBL3695219

COc1ccc(OC)c(C=CC(=O)c2ccccc2N(C)CCN(C)C)c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.59
PDE4B Q07343 1/20 0.59
PDE4C Q08493 1/20 0.59
PDE4D Q08499 1/20 0.59
ABCG2 Q9UNQ0 2/20 0.55
PTPN1 P18031 2/20 0.52
JUN P05412 1/20 0.52
NFKB1 P19838 1/20 0.52
MAPT P10636 3/20 0.50
LMNA P02545 2/20 0.50
ATM Q13315 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
GAA P10253 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAOB P27338 1/20 0.48
TNFRSF1A P19438 1/20 0.48
APP P05067 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690295 0.92 MAPT (0.60) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3685698 0.88 AR (0.60) PTPN1MAPTLMNAKDM4EMAOB
SCHEMBL3686633 0.88 AR (0.60) PTPN1MAPTLMNAKDM4EMAOB
SCHEMBL3695218 0.87 MAPT (0.59) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL6050485 0.87 MAPT (0.59) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3686915 0.86 MAOB (0.46) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3682205 0.86 MAOB (0.46) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3690293 0.85 ABCG2 (0.62) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3694613 0.85 ABCG2 (0.62) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3691412 0.84 ABCG2 (0.54) ABCG2PTPN1LMNASMN1; SMN2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed