SCHEMBL3696324

SCHEMBL3696324

Cc1ccc(F)c(-n2nc(CN(C)C(=O)OC(C)(C)C)cc2S(=O)(=O)c2ccc(Cl)nc2)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.40
SLC6A4 P31645 8/20 0.40
HTR2A P28223 1/20 0.39
KAT6A Q92794 1/20 0.32
KAT5 Q92993 1/20 0.32
KDM4E B2RXH2 1/20 0.31
RORC P51449 1/20 0.31
ALDH1A1 P00352 3/20 0.31
CYP2D6 P10635 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
RXRA P19793 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30
F2 P00734 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700225 0.94 HTR2C (0.39) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3700978 0.93 HTR2C (0.45) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3698587 0.90 HTR2C (0.42) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3697673 0.89 HTR2C (0.39) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL4131270 0.88 ALDH1A1 (0.37) KDM4EALDH1A1CYP2D6MEN1KMT2A
SCHEMBL3705902 0.87 HTR2C (0.39) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3703585 0.87 HTR2C (0.41) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3700004 0.87 HTR2C (0.39) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3814403 0.87 HTR2C (0.38) HTR2CSLC6A4HTR2AKAT6AKAT5
SCHEMBL3698341 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2AF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed