SCHEMBL3697127

SCHEMBL3697127

COc1ccc2nccc(CN[N+]3(N(C(=O)[O-])C(C)(C)C)CCCCCC3)c2c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.48
MTNR1B P49286 3/20 0.48
ROCK2 O75116 1/20 0.46
LMNA P02545 1/20 0.42
KDM4E B2RXH2 2/20 0.41
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP1A2 P05177 1/20 0.40
SLC22A12 Q96S37 1/20 0.39
KCNH2 Q12809 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5651810 0.82 MTNR1A (0.50) MTNR1AMTNR1BROCK2LMNAKDM4E
SCHEMBL5651807 0.70 MTNR1A (0.50) MTNR1AMTNR1BROCK2LMNAKDM4E
SCHEMBL3688184 0.69 ROCK2 (0.54) MTNR1AMTNR1BROCK2LMNAKDM4E
SCHEMBL3690391 0.68 KCNH2 (0.49) MTNR1AMTNR1BROCK2LMNAKCNH2
SCHEMBL4081621 0.68 MTNR1A (0.64) MTNR1AMTNR1BROCK2LMNAKDM4E
SCHEMBL12776123 0.67 MTNR1A (0.55) MTNR1AMTNR1BROCK2LMNAKDM4E
SCHEMBL13145890 0.67 KCNH2 (0.49) MTNR1AMTNR1BKCNH2
SCHEMBL2544860 0.67 MTNR1A (0.61) MTNR1AMTNR1BROCK2LMNAKDM4E
SCHEMBL5651333 0.66 KCNH2 (0.48) MTNR1AMTNR1BROCK2KCNH2
Bromide SCHEMBL30402372 0.66 MTNR1A (0.60) MTNR1AMTNR1BROCK2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed
EP-1551829-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2005-07-13 EP disclosed
WO-2004035569-A2 NOVEL COMPOUNDS WITH ANTIBACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2004-04-29 WO disclosed