SCHEMBL3697997

SCHEMBL3697997

CN(Cc1cc(S(=O)(=O)c2ccccc2)n(-c2cccnc2F)n1)C(=O)OC(C)(C)C.COc1ncccc1-n1nc(CN(C)C(=O)OC(C)(C)C)cc1S(=O)(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.41
SLC6A4 P31645 7/20 0.41
HTR2A P28223 1/20 0.38
SLC16A3 O15427 5/20 0.33
SLC16A1 P53985 5/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
F2 P00734 2/20 0.33
P2RX7 Q99572 1/20 0.33
NR1I2 O75469 1/20 0.32
AAK1 Q2M2I8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3697758 0.96 HTR2C (0.43) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL3700738 0.94 HTR2C (0.44) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL476325 0.88 HTR2C (0.42) HTR2CSLC6A4HTR2A
SCHEMBL3705968 0.88 SLC16A3 (0.39) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL3807718 0.87 HTR2C (0.41) HTR2CSLC6A4HTR2A
SCHEMBL476414 0.86 HTR2C (0.39) HTR2CSLC6A4HTR2AF2
SCHEMBL4131220 0.86 SMO (0.35) SLC16A3SLC16A1P2RX7NR1I2
SCHEMBL476337 0.85 HTR2C (0.38) HTR2CSLC6A4HTR2AF2
SCHEMBL3697999 0.85 P2RX7 (0.33) SLC16A3SLC16A1MMP2MMP9MMP8
SCHEMBL476394 0.83 HTR2C (0.37) HTR2CSLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed