SCHEMBL3699809

SCHEMBL3699809

Cc1c(F)cccc1-n1nc(CC(NC(=O)O)C(C)(C)C)cc1S(=O)(=O)c1cccnc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR1 P21462 1/20 0.39
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
NAMPT P43490 6/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
PTGER2 P43116 2/20 0.32
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
CACNA1G O43497 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3695803 0.94 FPR1 (0.38) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3808568 0.94 FPR1 (0.39) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL4566346 0.90 FPR1 (0.38) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3701317 0.89 FPR1 (0.38) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3693159 0.89 FPR1 (0.42) FPR1ABCC9ABCC8KCNJ11KCNJ8
Hydrochloric Acid SCHEMBL3707038 0.89 FPR1 (0.36) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3705290 0.86 FPR1 (0.41) FPR1ABCC9ABCC8KCNJ11KCNJ8
Fumaric Acid SCHEMBL3705163 0.85 FPR1 (0.33) FPR1ABCC9ABCC8KCNJ11KCNJ8
Fumaric Acid SCHEMBL3705157 0.85 FPR1 (0.33) FPR1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3697138 0.85 SLC16A3 (0.34) ABCC9ABCC8KCNJ11KCNJ8CACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed