SCHEMBL370029

SCHEMBL370029

O=C(O)c1cnc(-c2cccnc2)o1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
KDM4E B2RXH2 3/20 0.59
HPGD P15428 2/20 0.59
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
HSD17B10 Q99714 1/20 0.59
PIM1 P11309 1/20 0.52
PIM2 Q9P1W9 1/20 0.52
MKNK1 Q9BUB5 2/20 0.50
MKNK2 Q9HBH9 2/20 0.50
F2 P00734 1/20 0.49
IKBKB O14920 1/20 0.48
KMO O15229 2/20 0.48
CES1 P23141 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
EGFR P00533 1/20 0.46
PTGS2 P35354 1/20 0.46
FAAH O00519 1/20 0.45
APP P05067 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27790042 0.89 ALDH1A1 (0.57) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL2007486 0.84 CES1 (0.56) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL2116553 0.82 KDM4E (0.50) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL364612 0.79 ALDH1A1 (0.62) ALDH1A1HPGDNPC1RAB9APIM1
SCHEMBL17212184 0.79 HCAR2 (0.43) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL22436921 0.79 KDM4E (0.52) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL29505525 0.77 SMN1; SMN2 (0.47) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL16703005 0.77 CES1 (0.54) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL16896358 0.77 SMN1; SMN2 (0.47) ALDH1A1KDM4EHPGDNPC1RAB9A
SCHEMBL370030 0.77 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
EP-2593447-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-05-22 EP disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
WO-2012007500-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-01-19 WO disclosed
WO-2012007500-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides DDT, PTMS, ACHE ALDH1A1 2531/4885KDM4E 1038/4885HPGD 853/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.