SCHEMBL3701689

SCHEMBL3701689

Cc1ccccc1-c1cccc(C(N)=O)c1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.51
BCAT2 O15382 1/20 0.47
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
IKBKB O14920 1/20 0.45
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
BRD4 O60885 1/20 0.43
KDM4E B2RXH2 2/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GRK6 P43250 1/20 0.41
JAK2 O60674 1/20 0.41
MAPK14 Q16539 1/20 0.40
PARP1 P09874 2/20 0.40
BTK Q06187 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1512155 0.87 BCAT2 (0.55) MYCBCAT2KEAP1NFE2L2IKBKB
SCHEMBL3824312 0.86 MYC (0.66) MYCALDH1A1HPGDLMNAL3MBTL1
SCHEMBL1788703 0.85 BCAT2 (0.59) MYCBCAT2KEAP1NFE2L2IKBKB
SCHEMBL3135445 0.84 MYC (0.53) MYCBCAT2KEAP1NFE2L2IKBKB
SCHEMBL5742619 0.84 MYC (0.53) MYCBCAT2KEAP1NFE2L2IKBKB
SCHEMBL158431 0.83 CD44 (0.48) MYCBCAT2ALDH1A1HPGDLMNA
SCHEMBL29442190 0.83 CD44 (0.48) MYCBCAT2ALDH1A1HPGDLMNA
SCHEMBL28471957 0.81 MYC (0.59) MYCBCAT2KEAP1NFE2L2IKBKB
SCHEMBL3804575 0.81 ALDH1A1 (0.50) BCAT2KEAP1NFE2L2IKBKBALDH1A1
SCHEMBL4138458 0.79 MYC (0.72) MYCBCAT2KEAP1NFE2L2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed