SCHEMBL3701694

SCHEMBL3701694

Cc1c(-c2ccccc2)ccc(N)c1C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.46
IKBKB O14920 3/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
GAA P10253 1/20 0.44
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
MAP2K3 P46734 1/20 0.42
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 2/20 0.41
USP2 O75604 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
RECQL P46063 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4671318 0.88 PDE4A (0.44) BCAT2IKBKBMEN1KMT2APDE4A
SCHEMBL3135452 0.84 BCAT2 (0.47) BCAT2MEN1KMT2AGAAALDH1A1
Hydrochloric Acid SCHEMBL29287793 0.83 CA1 (0.47) BCAT2MEN1KMT2AGAAALDH1A1
Hydrochloric Acid SCHEMBL29287828 0.83 CA1 (0.47) BCAT2MEN1KMT2AGAAALDH1A1
SCHEMBL17829925 0.77 BCAT2 (0.56) BCAT2IKBKBMEN1KMT2AALDH1A1
SCHEMBL1250167 0.77 BCAT2 (0.55) BCAT2IKBKBMEN1KMT2AGAA
SCHEMBL31255442 0.76 BCAT2 (0.42) BCAT2IKBKBMEN1KMT2AGAA
SCHEMBL27824725 0.76 CHEK2 (0.50) BCAT2IKBKBMEN1KMT2AGAA
SCHEMBL3698514 0.75 FABP4 (0.40) BCAT2IKBKBMEN1KMT2AGAA
SCHEMBL141445 0.75 HSD17B10 (0.50) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed