SCHEMBL370210

SCHEMBL370210

Cc1ccc(C(CC(=NO)C2=CC=CN(C)C2)c2ccc(-c3ccc(C(=O)O)cc3)cc2)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.43
KDM4E B2RXH2 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
ADRB3 P13945 1/20 0.30
MRGPRX4 Q96LA9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370503 0.85 GPBAR1 (0.46) GPBAR1RXRARXRBADRB3
SCHEMBL1390243 0.79 GPBAR1 (0.47) GPBAR1KDM4ERXRARXRBADRB3
SCHEMBL1390242 0.79 GPBAR1 (0.47) GPBAR1KDM4ERXRARXRBADRB3
SCHEMBL1390240 0.79 GPBAR1 (0.47) GPBAR1KDM4ERXRARXRBADRB3
SCHEMBL370694 0.76 GPBAR1 (0.37) GPBAR1KDM4E
SCHEMBL362457 0.75 GPBAR1 (0.48) GPBAR1KDM4ERXRARXRB
SCHEMBL1389996 0.71 GPBAR1 (0.45) GPBAR1KDM4ERXRARXRB
SCHEMBL370196 0.71 GPBAR1 (0.42) GPBAR1
SCHEMBL1390000 0.71 GPBAR1 (0.45) GPBAR1KDM4ERXRARXRB
SCHEMBL15949194 0.71 GPBAR1 (0.38) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed