SCHEMBL370503

SCHEMBL370503

Cc1cc(Cl)ccc1C(CC(=NO)C1=CC=CN(C)C1)c1ccc(-c2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.46
PPARG P37231 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
SRD5A2 P31213 1/20 0.31
PTGER4 P35408 2/20 0.31
PTGER2 P43116 2/20 0.31
PTGER1 P34995 1/20 0.31
PTGER3 P43115 1/20 0.31
HSD11B1 P28845 1/20 0.31
PHGDH O43175 1/20 0.31
ADRB1 P08588 3/20 0.31
ADRB3 P13945 3/20 0.31
PLA2G4A P47712 2/20 0.31
RXRA P19793 2/20 0.31
RXRB P28702 1/20 0.31
GRM1 Q13255 2/20 0.30
MEN1 O00255 1/20 0.30
CYP1A2 P05177 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370694 0.90 GPBAR1 (0.37) GPBAR1PPARGKEAP1NFE2L2MEN1
SCHEMBL370210 0.85 GPBAR1 (0.43) GPBAR1ADRB3RXRARXRB
SCHEMBL369177 0.84 GPBAR1 (0.33) GPBAR1KEAP1NFE2L2
SCHEMBL369976 0.83 GPBAR1 (0.35) GPBAR1
SCHEMBL369931 0.79 GPBAR1 (0.51) GPBAR1PPARGKEAP1NFE2L2SRD5A2
SCHEMBL1390130 0.79 GPBAR1 (0.51) GPBAR1PPARGKEAP1NFE2L2SRD5A2
SCHEMBL10241339 0.79 GPBAR1 (0.51) GPBAR1PPARGKEAP1NFE2L2SRD5A2
SCHEMBL369930 0.79 GPBAR1 (0.51) GPBAR1PPARGKEAP1NFE2L2SRD5A2
SCHEMBL10241335 0.79 GPBAR1 (0.51) GPBAR1PPARGKEAP1NFE2L2SRD5A2
SCHEMBL370370 0.78 FFAR1 (0.33) PTGER4PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed