SCHEMBL370694

SCHEMBL370694

Cc1cc(Cl)ccc1C(CC(=NO)C1=CC=CN(C)C1)c1ccc(-c2ccc(C(=O)NCC(=O)O)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.37
GCG P01275 2/20 0.34
PPARG P37231 1/20 0.33
EGLN1 Q9GZT9 3/20 0.32
VEGFA P15692 2/20 0.32
FLT1 P17948 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
GCGR P47871 3/20 0.31
ADCY6 O43306 1/20 0.31
ADCY3 O60266 1/20 0.31
ADCY9 O60503 1/20 0.31
ADCY5 O95622 1/20 0.31
ADCY8 P40145 1/20 0.31
ADCY7 P51828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370503 0.90 GPBAR1 (0.46) GPBAR1PPARGMEN1CYP1A2KMT2A
SCHEMBL369976 0.86 GPBAR1 (0.35) GPBAR1GCGALDH1A1GCGR
SCHEMBL1389730 0.81 GPBAR1 (0.41) GPBAR1GCGPPARGEGLN1VEGFA
SCHEMBL1389593 0.81 GPBAR1 (0.41) GPBAR1GCGPPARGEGLN1VEGFA
SCHEMBL1389596 0.81 GPBAR1 (0.41) GPBAR1GCGPPARGEGLN1VEGFA
SCHEMBL369177 0.80 GPBAR1 (0.33) GPBAR1KEAP1NFE2L2
SCHEMBL363289 0.78 GPBAR1 (0.41) GPBAR1GCGPPARGEGLN1VEGFA
SCHEMBL370210 0.76 GPBAR1 (0.43) GPBAR1KDM4E
SCHEMBL1389691 0.74 GPBAR1 (0.39) GPBAR1GCGPPARGEGLN1MEN1
SCHEMBL1389689 0.74 GPBAR1 (0.39) GPBAR1GCGPPARGEGLN1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed