SCHEMBL3702181

SCHEMBL3702181

Cc1ccc(S(=O)(=O)c2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2ccccc2Cl)nc1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 13/20 0.37
SLC16A1 P53985 12/20 0.37
TRPM8 Q7Z2W7 1/20 0.35
FPR1 P21462 1/20 0.33
PDE4B Q07343 1/20 0.33
GCK P35557 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
KCNH2 Q12809 1/20 0.32
CCR9 P51686 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696895 0.89 SLC16A3 (0.44) SLC16A3SLC16A1
SCHEMBL3700362 0.87 SLC16A3 (0.38) SLC16A3SLC16A1TRPM8FPR1PDE4B
SCHEMBL3696613 0.85 SLC16A3 (0.37) SLC16A3SLC16A1TRPM8FPR1PDE4B
SCHEMBL3701987 0.85 SLC16A3 (0.36) SLC16A3SLC16A1PDE4B
SCHEMBL3696908 0.84 ALDH1A1 (0.39) SLC16A3SLC16A1FPR1
SCHEMBL3701584 0.83 SLC16A3 (0.39) SLC16A3SLC16A1PDE4B
SCHEMBL3698141 0.83 SLC16A3 (0.37) SLC16A3SLC16A1TRPM8FPR1PDE4B
SCHEMBL3698156 0.82 KMT2A (0.38) SLC16A3SLC16A1
SCHEMBL3702179 0.82 HTR2C (0.43) SLC16A3SLC16A1
SCHEMBL3691770 0.82 SLC16A3 (0.40) SLC16A3SLC16A1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed