SCHEMBL3701987

SCHEMBL3701987

Cc1cccc(S(=O)(=O)c2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2ccccc2Cl)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 15/20 0.36
SLC16A1 P53985 14/20 0.36
PDE4B Q07343 1/20 0.34
RXRA P19793 2/20 0.32
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32
P2RY1 P47900 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
MITF O75030 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3691770 0.90 SLC16A3 (0.40) SLC16A3SLC16A1PDE4BRXRANR1H2
SCHEMBL3696895 0.88 SLC16A3 (0.44) SLC16A3SLC16A1KDM4E
SCHEMBL4118797 0.86 SLC16A3 (0.36) SLC16A3SLC16A1PDE4BKDM4EMEN1
SCHEMBL3702181 0.85 SLC16A3 (0.37) SLC16A3SLC16A1PDE4B
SCHEMBL3696613 0.84 SLC16A3 (0.37) SLC16A3SLC16A1PDE4BP2RY1ALDH1A1
SCHEMBL3701584 0.84 SLC16A3 (0.39) SLC16A3SLC16A1PDE4BRXRANR1H2
SCHEMBL3696908 0.82 ALDH1A1 (0.39) SLC16A3SLC16A1MEN1ALDH1A1KMT2A
SCHEMBL3701985 0.82 HTR2C (0.43) SLC16A3SLC16A1PDE4B
SCHEMBL4201755 0.81 SLC16A3 (0.36) SLC16A3SLC16A1PDE4BP2RY1MEN1
SCHEMBL3698156 0.80 KMT2A (0.38) SLC16A3SLC16A1RXRANR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed