SCHEMBL3702610

SCHEMBL3702610

CCS(=O)(=O)c1ccc(-c2ccc([C@@H](C#N)CNC(=O)C3CCCCN3C(=O)O)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSC P53634 3/20 0.41
FKBP1A P62942 5/20 0.39
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 1/20 0.35
CTSK P43235 2/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
KMT2A Q03164 1/20 0.35
FKBP5 Q13451 1/20 0.35
XIAP P98170 1/20 0.34
MLX Q9UH92 1/20 0.34
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP13 P45452 1/20 0.34
ADAM17 P78536 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3688512 0.86 CTSC (0.41) CTSCFKBP1AKMT2AFKBP5XIAP
SCHEMBL3662346 0.85 KMT2A (0.45) FKBP1ANPC1SMN1; SMN2MMP2MMP9
SCHEMBL3661348 0.83 FKBP1A (0.39) FKBP1ANPC1CTSKKMT2AFKBP5
SCHEMBL3656005 0.80 CTSC (0.42) CTSCCTSK
SCHEMBL16478103 0.79 CTSC (0.41) CTSCCTSK
SCHEMBL3657032 0.78 CTSC (0.49) CTSCCTSK
SCHEMBL3659109 0.77 FKBP1A (0.36) FKBP1ATDP1KMT2AFKBP5XIAP
SCHEMBL3657671 0.74 CTSC (0.44) CTSCMMP13
SCHEMBL3692633 0.73 VHL (0.57) XIAP
SCHEMBL1499091 0.73 CTSC (0.37) CTSCMAPTTDP1SMN1; SMN2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010142985-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL]PIPERIDIN-2-YLCARBOXMIDE COMPOUNDS 761 ASTRAZENECA AB (SE) 2010-12-16 WO disclosed