SCHEMBL3703586

SCHEMBL3703586

Cc1ccc(F)cc1-n1nc(CN(CC(C)(C)C)C(=O)O)cc1S(=O)(=O)c1ccc(Cl)nc1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
THRB P10828 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TRPA1 O75762 4/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
CYP2D6 P10635 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
KCNH2 Q12809 1/20 0.31
RORC P51449 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700979 0.93 KCNQ3 (0.34) ALDH1A1THRBMEN1KMT2AKCNQ3
SCHEMBL3814411 0.88 ALDH1A1 (0.34) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL4130773 0.88 ALDH1A1 (0.37) ALDH1A1THRBMEN1KMT2AKCNQ3
SCHEMBL3697103 0.87 PRCP (0.33) TRPA1HTR2AHTR2CKCNH2TRPM8
SCHEMBL3697675 0.87 ALDH1A1 (0.35) ALDH1A1MEN1KMT2AKCNQ3KCNQ2
SCHEMBL3696326 0.87 ALDH1A1 (0.33) ALDH1A1MEN1KMT2AKCNQ3KCNQ2
SCHEMBL3700226 0.87 ALDH1A1 (0.33) ALDH1A1THRBMEN1KMT2AKCNQ3
SCHEMBL3698589 0.87 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AKCNQ3KCNQ2
SCHEMBL3706787 0.86 CNR1 (0.32) ALDH1A1THRBMEN1KMT2AKCNQ3
SCHEMBL3705903 0.85 ALDH1A1 (0.35) ALDH1A1MEN1KMT2AKCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed