SCHEMBL3697103

SCHEMBL3697103

Cc1ccc(S(=O)(=O)c2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2cc(F)ccc2Cl)cn1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRCP P42785 2/20 0.33
P2RX7 Q99572 2/20 0.32
TRPA1 O75762 1/20 0.31
PTGDR2 Q9Y5Y4 4/20 0.31
PTGDR Q13258 2/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696613 0.89 SLC16A3 (0.37) TRPM8
SCHEMBL3705296 0.89 NAMPT (0.34) PTGDR2
SCHEMBL3688572 0.88 RIPK1 (0.34) TRPM8
SCHEMBL3704890 0.88 P2RX7 (0.34) PRCPP2RX7PTGDR2PTGDRTRPM8
SCHEMBL3703586 0.87 ALDH1A1 (0.33) TRPA1TRPM8HTR2AHTR2CKCNH2
SCHEMBL3700979 0.86 KCNQ3 (0.34) TRPA1HTR2AHTR2CKCNH2
SCHEMBL3700610 0.86 SLC16A3 (0.33) HTR2AHTR2CKCNH2
SCHEMBL3706787 0.86 CNR1 (0.32)
SCHEMBL3700701 0.85 RXRA (0.32) HTR2AHTR2CKCNH2
SCHEMBL3698342 0.85 NAMPT (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed