SCHEMBL3704969

SCHEMBL3704969

CC(=N)C(Nc1ccc2oc(C3=COC(Cc4ccccc4)O3)c(O)c(=O)c2c1)C1CC1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
MAPT P10636 1/20 0.35
VKORC1 Q9BQB6 2/20 0.30
MEN1 O00255 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
ABCB1 P08183 1/20 0.30
CYP3A4 P08684 1/20 0.30
CALM1 P0DP23 1/20 0.30
AR P10275 1/20 0.30
PKM P14618 1/20 0.30
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP1B1 Q16678 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL928102 0.89 ABCG2 (0.32) ABCB1
Hydrochloric Acid SCHEMBL926191 0.84 KDM4E (0.39) KDM4EMAPTMEN1CA12CA1
SCHEMBL926119 0.82 KDM4E (0.40) KDM4EMAPTMEN1CA12CA1
Hydrochloric Acid SCHEMBL926419 0.81 KDM4E (0.35) KDM4EMAPTMEN1CA12CA1
SCHEMBL7666892 0.80 SNCA (0.45) KDM4EMAPTMEN1LMNAKMT2A
SCHEMBL7662615 0.79 CA12 (0.38) KDM4EMAPTMEN1CA12CA1
SCHEMBL7666098 0.78 MAPT (0.58) KDM4EMAPTMEN1CA12CA1
SCHEMBL7654027 0.78 MAOA (0.37) KDM4EMAPTMEN1CA12KMT2A
SCHEMBL7664375 0.76 MAPT (0.43) KDM4EMAPTMEN1CA12TP53
SCHEMBL7656081 0.76 MAPT (0.48) KDM4EMAPTMEN1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268628-B1 2-ARYL AND 2 -HETEROARYL 4H-1-BENZOPYRAN-4-ONE-6-AMIDINO DERIVATIVES FOR THE TREATMENT OF ARTHRITIS, CANCER AND RELATED PAIN ROTTAPHARM SPA (IT) 2012-05-16 EP disclosed