SCHEMBL3708933

SCHEMBL3708933

Cc1ccccc1N1CCC(N2CCN(C(C)c3ccccc3)CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.53
CHRM2 P08172 8/20 0.50
CHRM1 P11229 7/20 0.50
OPRM1 P35372 2/20 0.48
OPRK1 P41145 1/20 0.48
OPRL1 P41146 1/20 0.48
MC4R P32245 1/20 0.48
L3MBTL3 Q96JM7 3/20 0.45
MBTD1 Q05BQ5 2/20 0.45
SLC18A3 Q16572 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.43
CCR5 P51681 2/20 0.43
TRPC5 Q9UL62 1/20 0.41
ADRB1 P08588 1/20 0.41
CHRM4 P08173 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3703903 0.99 CYP2D6 (0.51) CYP2D6CHRM2CHRM1OPRM1OPRK1
SCHEMBL3709196 0.95 OPRM1 (0.51) CYP2D6CHRM2CHRM1OPRM1OPRK1
Hydrochloric Acid SCHEMBL3808136 0.94 OPRM1 (0.50) CYP2D6CHRM2CHRM1OPRM1OPRK1
SCHEMBL13283844 0.87 CHRM2 (0.51) CYP2D6CHRM2CHRM1OPRM1OPRK1
SCHEMBL3703344 0.85 CHRM2 (0.51) CHRM2CHRM1OPRM1OPRK1OPRL1
Hydrochloric Acid SCHEMBL3708307 0.84 CHRM2 (0.50) CHRM2CHRM1OPRM1OPRK1OPRL1
SCHEMBL3714873 0.83 CHRM2 (0.54) CHRM2CHRM1OPRM1SLC18A3CHRM4
Hydrochloric Acid SCHEMBL3708326 0.82 CHRM2 (0.53) CHRM2CHRM1OPRM1SLC18A3CCR5
Hydrochloric Acid SCHEMBL3705110 0.81 SLC18A3 (0.41) CHRM2CHRM1OPRM1OPRK1OPRL1
SCHEMBL3708960 0.81 OPRM1 (0.43) CYP2D6CHRM2CHRM1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010081851-A1 PIPERIDIN-4-YLPIPERAZINE COMPOUNDS FOR THE TREATMENT OF HCV INFECTION GENOSCIENCE PHARMA (FR) 2010-07-22 WO disclosed
WO-2010081851-A1 PIPERIDIN-4-YLPIPERAZINE COMPOUNDS FOR THE TREATMENT OF HCV INFECTION GENOSCIENCE PHARMA (FR) 2010-07-22 WO disclosed