SCHEMBL3709730

SCHEMBL3709730

COC(=O)c1cc(-c2ccccc2)nc(-c2ccc(C#Cc3cccnc3)cc2)c1OC

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 3/20 0.44
MAPK1 P28482 1/20 0.42
DHODH Q02127 2/20 0.42
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ALDH1A1 P00352 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NR4A2 P43354 2/20 0.40
KDM4E B2RXH2 2/20 0.40
TP53 P04637 1/20 0.40
FFAR1 O14842 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HPGD P15428 1/20 0.39
XIAP P98170 1/20 0.39
BIRC2 Q13490 1/20 0.39
AAK1 Q2M2I8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709739 0.90 MEN1 (0.41) DHODHALDH1A1MEN1KMT2AKDM4E
SCHEMBL3713520 0.86 GRM5 (0.46) MAPK1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL13188472 0.86 MAPT (0.42) CYP19A1CYP11B1CYP11B2ALDH1A1MEN1
SCHEMBL3720782 0.86 MEN1 (0.47) MAPK1CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL3716537 0.86 MCL1 (0.47) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL3712449 0.84 GRM5 (0.44) MAPK1DHODHCYP11B1CYP11B2ALDH1A1
SCHEMBL13187704 0.83 NPC1 (0.44) CYP19A1CYP11B1CYP11B2ALDH1A1MEN1
SCHEMBL3713522 0.79 GRM5 (0.43) MAPK1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL3716967 0.79 ERN1 (0.46) KMT2ANR4A2KDM4EFFAR1AAK1
SCHEMBL3709575 0.79 ALDH1A1 (0.47) CYP19A1CYP11B1CYP11B2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed