SCHEMBL370976

SCHEMBL370976

COC(=O)c1ccc(-c2ccccc2)c(CCCc2ccccc2C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.50
PTGS2 P35354 1/20 0.48
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALOX12 P18054 1/20 0.47
SLC2A1 P11166 1/20 0.44
HTT P42858 1/20 0.42
CYP4A11 Q02928 3/20 0.41
CYP4F2 P78329 2/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
NEK1 Q96PY6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370894 0.87 RARB (0.46) EGFRMEN1KMT2ATSHRALDH1A1
SCHEMBL369805 0.85 CYP4A11 (0.50) EGFRPTGS2MEN1KMT2AALOX12
SCHEMBL4664597 0.81 EGFR (0.60) EGFRPTGS2MAPTMEN1KMT2A
SCHEMBL3748237 0.78 EGFR (0.63) EGFRPTGS2MAPTMEN1KMT2A
SCHEMBL27621631 0.78 EGFR (0.56) EGFRPTGS2MAPTMEN1KMT2A
SCHEMBL821283 0.75 PTGS2 (0.59) EGFRPTGS2MAPTMEN1KMT2A
SCHEMBL410454 0.75 EGFR (0.46) EGFRPTGS2MAPTMEN1KMT2A
SCHEMBL10458005 0.75 PTGS2 (0.76) EGFRPTGS2MAPTMEN1KMT2A
SCHEMBL11208106 0.74 TAAR1 (0.48) KMT2AALDH1A1LMNAL3MBTL1TDP1
SCHEMBL2771823 0.74 PTGS2 (0.59) EGFRPTGS2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed