SCHEMBL370983

SCHEMBL370983

Brc1cccc(-c2nnc(Nc3ccccc3)s2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.58
RAB9A P51151 7/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
HDAC6 Q9UBN7 1/20 0.53
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 1/20 0.50
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CB P42338 1/20 0.47
KDR P35968 1/20 0.46
ROCK1 Q13464 2/20 0.45
CSNK2A2 P19784 1/20 0.44
CSNK2B P67870 1/20 0.44
CSNK2A1 P68400 1/20 0.44
CSNK2A3 Q8NEV1 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
TP53 P04637 3/20 0.44
TSHR P16473 1/20 0.44
ROCK2 O75116 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23220346 0.89 NPC1 (0.67) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL12015939 0.84 NPC1 (0.73) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL6154268 0.83 HSD17B1 (0.58) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL28573293 0.83 HDAC6 (0.65) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL28593202 0.83 NPC1 (0.59) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL29367007 0.82 NPC1 (0.58) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL28593204 0.82 NPC1 (0.58) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL6154099 0.82 ROCK2 (0.62) NPC1RAB9AMEN1KMT2AHDAC6
SCHEMBL6153968 0.80 KDM4E (0.52) NPC1RAB9AMEN1KMT2AROCK1
SCHEMBL27879285 0.78 NPC1 (0.51) NPC1RAB9AMEN1KMT2AHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593106-A1 ORGANIC COMPOUNDS Rockefeller University (US) 2013-05-22 EP disclosed
WO-2012009688-A1 ORGANIC COMPOUNDS ROCKEFELLER UNIVERSITY (US) 2012-01-19 WO disclosed