SCHEMBL3709958

SCHEMBL3709958

CCCCC(=O)c1cc(Cl)ccc1OC(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 1/20 0.42
HTR2C P28335 3/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
F2R P25116 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP2D6 P10635 1/20 0.40
PKM P14618 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2B P41595 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28758200 0.86 ANO1 (0.45) ANO1ALDH1A1KDM4ELMNACYP11B1
SCHEMBL3922656 0.80 ANO1 (0.42) ANO1HTR2CLMNACYP11B1CYP11B2
SCHEMBL29648921 0.78 ANO1 (0.46) ANO1KDM4ELMNACYP1A2CYP3A4
SCHEMBL22979877 0.78 ANO1 (0.46) ANO1KDM4ELMNACYP1A2CYP3A4
SCHEMBL29646503 0.76 TSHR (0.53) ANO1ALDH1A1L3MBTL1CYP11B1CYP11B2
SCHEMBL2115556 0.76 TSHR (0.53) ANO1ALDH1A1L3MBTL1CYP11B1CYP11B2
SCHEMBL30843111 0.76 ABL1 (0.51) ANO1ALDH1A1LMNAMEN1KMT2A
SCHEMBL8712803 0.75 HTT (0.54) ALDH1A1KDM4ELMNATDP1MEN1
SCHEMBL31743138 0.75 MAP2 (0.50) ANO1ALDH1A1KDM4ECYP11B1CYP11B2
SCHEMBL16957723 0.75 ANO1 (0.44) ANO1HTR2CALDH1A1LMNACYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398796-A1 HETEROCYCLIC DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Canada Inc. (CA) 2011-12-28 EP disclosed
WO-2010094126-A1 HETEROCYCLIC DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-08-26 WO disclosed