SCHEMBL3711230

SCHEMBL3711230

COC(=O)c1cc(C#Cc2cccnc2)cnc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.46
ALDH1A1 P00352 2/20 0.46
CSF1R P07333 1/20 0.44
AAK1 Q2M2I8 1/20 0.44
KDM4E B2RXH2 4/20 0.44
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 2/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
GRM5 P41594 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
CYP2A6 P11509 1/20 0.40
CYP2C9 P11712 1/20 0.40
CHRNB2 P17787 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40
CHRNA4 P43681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188251 0.88 CSF1R (0.45) ERN1CSF1RAAK1KDM4EPTGDR2
SCHEMBL3711387 0.87 AAK1 (0.45) ERN1ALDH1A1CSF1RAAK1KDM4E
SCHEMBL3711323 0.85 AAK1 (0.45) ERN1ALDH1A1CSF1RAAK1KDM4E
SCHEMBL3711431 0.80 CSF1R (0.53) ERN1ALDH1A1CSF1RAAK1KDM4E
SCHEMBL25294855 0.80 ALDH1A1 (0.51) ERN1ALDH1A1CSF1RAAK1PTGDR2
SCHEMBL3711926 0.79 ALDH1A1 (0.44) ERN1ALDH1A1CSF1RAAK1KDM4E
SCHEMBL3714223 0.79 ALDH1A1 (0.62) ERN1ALDH1A1CSF1RKDM4EKMT2A
SCHEMBL3714907 0.78 MAPT (0.50) ALDH1A1
SCHEMBL5781938 0.77 NR4A2 (0.54) ALDH1A1KDM4EGABRA1GABRG2GABRB3
SCHEMBL26101255 0.77 ALDH1A1 (0.40) ALDH1A1KDM4EGRM5CYP2C9CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed