SCHEMBL3714907

SCHEMBL3714907

COC(=O)c1cc(C#Cc2cccnc2)cnc1N1CCOCC1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.50
PIK3CA P42336 10/20 0.47
OPRK1 P41145 3/20 0.46
ALDH1A1 P00352 1/20 0.44
PLOD2 O00469 1/20 0.43
PLOD3 O60568 1/20 0.43
PLOD1 Q02809 1/20 0.43
MTOR P42345 1/20 0.42
LRRK2 Q5S007 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188148 0.87 PIK3CA (0.46) MAPTPIK3CAPLOD2PLOD3PLOD1
SCHEMBL17478867 0.80 ALDH1A1 (0.60) OPRK1ALDH1A1LRRK2
SCHEMBL3715549 0.79 OPRK1 (0.44) OPRK1ALDH1A1
SCHEMBL3711230 0.78 ERN1 (0.46) ALDH1A1
SCHEMBL16105029 0.76 OPRK1 (0.61) MAPTOPRK1ALDH1A1
SCHEMBL3711323 0.76 AAK1 (0.45) ALDH1A1
SCHEMBL3713658 0.75 OPRK1 (0.40) OPRK1
SCHEMBL3719404 0.74 OPRK1 (0.75) OPRK1
SCHEMBL29574379 0.74 OPRK1 (0.75) OPRK1
SCHEMBL3714505 0.73 PIK3CA (0.48) MAPTPIK3CAPLOD2PLOD3PLOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed