SCHEMBL3711255

SCHEMBL3711255

COC(=O)[C@H](COCC1(C)CC1)NC(=O)C1(c2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
UGCG Q16739 17/20 0.54
CYP3A4 P08684 15/20 0.54
ALDH1A1 P00352 1/20 0.37
P2RX7 Q99572 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3712562 0.87 UGCG (0.54) UGCGCYP3A4ALDH1A1P2RX7
SCHEMBL13260342 0.85 UGCG (0.75) UGCGCYP3A4
SCHEMBL3805632 0.79 UGCG (0.55) UGCGCYP3A4P2RX7
SCHEMBL3719782 0.74 UGCG (0.41) UGCGCYP3A4ALDH1A1P2RX7
SCHEMBL21326254 0.72 UGCG (0.92) UGCGCYP3A4
SCHEMBL13260343 0.72 UGCG (0.92) UGCGCYP3A4
SCHEMBL13260406 0.71 UGCG (0.56) UGCGCYP3A4ALDH1A1
SCHEMBL3715484 0.71 UGCG (0.69) UGCGCYP3A4
SCHEMBL3709194 0.71 UGCG (0.69) UGCGCYP3A4
SCHEMBL13260997 0.70 UGCG (0.68) UGCGCYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010091164-A1 INHIBITORS OF GLUCOSYLCERAMIDE SYNTHASE EXELIXIS, INC. (US) 2010-08-12 WO disclosed