SCHEMBL3711802

SCHEMBL3711802

O=C1COCCN1C1CCCNC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
HTR2B P41595 7/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR3A P46098 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35
HTR6 P50406 1/20 0.35
HTR2C P28335 6/20 0.33
HTR2A P28223 3/20 0.33
PIK3CD O00329 4/20 0.32
PIK3CA P42336 4/20 0.32
PIK3CB P42338 4/20 0.32
PIK3R2 O00459 3/20 0.32
PIK3CG P48736 3/20 0.32
PIK3R5 Q8WYR1 3/20 0.32
PIK3R3 Q92569 3/20 0.32
NAAA Q02083 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21040531 0.84 HTR2C (0.39) HTR2BHTR2CHTR2A
SCHEMBL23187488 0.83 F10 (0.32) PIK3CD
SCHEMBL15972321 0.81 DGAT1 (0.38) PIK3CDMAPK1
SCHEMBL1976258 0.80 F10 (0.35) PARP1HTR2BHTR2CHTR2APIK3CD
SCHEMBL7886958 0.80 MEN1 (0.39) MAPK1
Hydrochloric Acid SCHEMBL3565110 0.79 F10 (0.34) PARP1HTR2BHTR2CHTR2APIK3CD
SCHEMBL29333188 0.78 NAAA (0.44) PARP1HTR2BHTR3EHTR3BHTR3A
SCHEMBL29332336 0.78 NAAA (0.44) PARP1HTR2BHTR3EHTR3BHTR3A
SCHEMBL29865291 0.77 F10 (0.38) PIK3CDIRAK4
SCHEMBL24710626 0.77 HTR2C (0.41) PARP1HTR2BHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010091721-A1 3 -SUBSTITUTED 1-ARYLSULFONYLPIPERIDINE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LIMITED (GB) 2010-08-19 WO disclosed
WO-2010091721-A1 3 -SUBSTITUTED 1-ARYLSULFONYLPIPERIDINE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LIMITED (GB) 2010-08-19 WO disclosed