SCHEMBL3712432

SCHEMBL3712432

COC(=O)c1cc(OCCN2CCOCC2)nc(-c2ccc(C#Cc3ccc(CN4CCOCC4)cc3)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.47
MAPK1 P28482 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM1A O60341 1/20 0.45
HDAC1 Q13547 1/20 0.45
KMT2A Q03164 1/20 0.43
BCHE P06276 1/20 0.42
MAOA P21397 1/20 0.42
ACHE P22303 1/20 0.42
MAOB P27338 1/20 0.42
ITK Q08881 1/20 0.42
ACP1 P24666 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720719 0.90 KMO (0.45) ACACBKDM1AHDAC1BCHEMAOA
SCHEMBL13187705 0.90 HDAC1 (0.55) ACACBKDM1AHDAC1
SCHEMBL13187744 0.88 HDAC1 (0.51) KDM1AHDAC1
SCHEMBL3712071 0.87 GAA (0.46) ACACBSMN1; SMN2KDM1AHDAC1BCHE
SCHEMBL3717935 0.86 MAPK1 (0.50) MAPK1SMN1; SMN2KMT2AACP1
SCHEMBL13187707 0.85 HDAC1 (0.48) KDM1AHDAC1KMT2A
SCHEMBL3713318 0.85 KMT2A (0.46) MAPK1SMN1; SMN2KMT2AITKACP1
SCHEMBL3711313 0.85 MAPK1 (0.49) MAPK1SMN1; SMN2KMT2AACP1
SCHEMBL3720383 0.84 AURKA (0.46) ACACBMAPK1SMN1; SMN2KMT2AACP1
SCHEMBL3710611 0.84 ACACB (0.47) ACACBMAPK1SMN1; SMN2KDM1AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed