SCHEMBL3712978

SCHEMBL3712978

CS(=O)(=O)c1cccc(-c2ccc3nc(NC(=O)C(=O)O)sc3c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.59
RAB9A P51151 7/20 0.59
PIK3CG P48736 1/20 0.59
ALDH1A1 P00352 6/20 0.56
MEN1 O00255 6/20 0.56
KMT2A Q03164 6/20 0.56
HSD17B10 Q99714 1/20 0.56
GAA P10253 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
KDM4E B2RXH2 3/20 0.55
RXFP1 Q9HBX9 2/20 0.55
ACP1 P24666 1/20 0.55
CLK1 P49759 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
ABL1 P00519 1/20 0.54
LMNA P02545 2/20 0.53
TP53 P04637 1/20 0.53
PKM P14618 1/20 0.53
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3710470 0.91 NPC1 (0.61) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL3869295 0.89 PIK3CG (0.72) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL13188645 0.86 ACP1 (0.62) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL13188200 0.86 PTPN1 (0.64) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL3919385 0.85 CLK1 (0.53) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL13188971 0.85 CLK1 (0.53) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL13189072 0.84 ALDH1A1 (0.81) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL3711380 0.81 NPC1 (0.49) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL3705975 0.81 ABL1 (0.59) NPC1RAB9APIK3CGALDH1A1MEN1
SCHEMBL13188972 0.81 RAB9A (0.81) NPC1RAB9AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed
WO-2009133127-A1 FUSED BICYCLIC COMPOUNDS AND USE THEREOF AS PI3K INHIBITORS MERCK SERONO S.A. (CH) 2009-11-05 WO disclosed