SCHEMBL3713383

SCHEMBL3713383

COC(=O)c1cc(-c2ccc(C#Cc3cccnc3)cc2)nc(N2CCC(OC)CC2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2D6 P10635 3/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP1A2 P05177 1/20 0.38
HRH3 Q9Y5N1 2/20 0.37
PAX8 Q06710 1/20 0.37
CDC7 O00311 1/20 0.37
DBF4 Q9UBU7 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
HIF1A Q16665 1/20 0.36
EPAS1 Q99814 1/20 0.36
PTGER4 P35408 1/20 0.36
CSF1R P07333 1/20 0.36
P2RY12 Q9H244 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714675 0.92 PTGER4 (0.42) CYP3A4CYP2D6CYP2C9CYP2C19CYP1A2
SCHEMBL3713715 0.91 CYP19A1 (0.40) CYP19A1CYP11B1CYP11B2PAX8ALDH1A1
SCHEMBL3711841 0.90 CYP19A1 (0.42) CYP19A1CYP11B1CYP11B2ALDH1A1HIF1A
SCHEMBL3711328 0.90 AIMP2 (0.39) CYP19A1CYP11B1CYP11B2PAX8ALDH1A1
SCHEMBL3711913 0.89 CYP19A1 (0.41) CYP19A1CYP11B1CYP11B2ALDH1A1HIF1A
SCHEMBL3712077 0.89 ABL1 (0.39) CYP19A1CYP11B1CYP11B2CYP3A4CYP2D6
SCHEMBL3709548 0.88 ALDH1A1 (0.42) CYP19A1CYP11B1CYP11B2CYP3A4CYP2D6
SCHEMBL13188255 0.88 CYP11B1 (0.49) CYP19A1CYP11B1CYP11B2CYP3A4CYP2D6
SCHEMBL3711200 0.88 PRKD1 (0.41) CYP19A1CYP11B1CYP11B2PAX8HIF1A
SCHEMBL3714505 0.88 PIK3CA (0.48) CYP19A1CYP11B1CYP11B2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed