SCHEMBL3714219

SCHEMBL3714219

[c]1[nH]c(-c2ccccc2)c(-c2ccco2)c1-c1cccs1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 1/20 0.43
ALDH1A1 P00352 9/20 0.41
KDM4E B2RXH2 7/20 0.41
HPGD P15428 6/20 0.41
HSD17B10 Q99714 4/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
MAPT P10636 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PPARG P37231 1/20 0.37
NCOA2 Q15596 1/20 0.37
NCOA1 Q15788 1/20 0.37
POLB P06746 2/20 0.36
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29696576 0.72 ALDH1A1 (0.54) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL5567841 0.69 ALDH1A1 (0.46) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL28741694 0.68 ALDH1A1 (0.51) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL521943 0.68 ALDH1A1 (0.62) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL745227 0.66 ALDH1A1 (0.46) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL28079025 0.63 ALDH1A1 (0.49) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL22733867 0.63 ALDH1A1 (0.49) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL18671634 0.62 ALDH1A1 (0.51) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3087312 0.62 ALDH1A1 (0.54) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL28253382 0.61 ESR1 (0.62) ALDH1A1KDM4EHPGDKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010077589-A2 STAT3 INHIBITORS AND THERAPEUTIC METHODS USING THE SAME THE REGENTS OF THE UNIVERSITY OF MICHIGAN OFFICE OF TECHNOLOGY TRANSFER (US) 2010-07-08 WO disclosed