SCHEMBL371457

SCHEMBL371457

[CH2]CC(C)C(N)=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852452 0.78
SCHEMBL7306532 0.78 CA1 (0.34)
SCHEMBL9611232 0.75 GABRR1 (0.38)
SCHEMBL2557939 0.74 LAP3 (0.35)
SCHEMBL3803892 0.74
SCHEMBL24433790 0.73
SCHEMBL131165 0.73
SCHEMBL308592 0.73
SCHEMBL16123655 0.73
SCHEMBL128376 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 175 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240116979-A1 METHOD FOR PRODUCING LIPIDIC PEPTIDE NISSAN CHEMICAL CORPORATION (JP) 2024-04-11 US claimed
US-20240067675-A1 METHOD FOR PRODUCING LIPID PEPTIDE NISSAN CHEMICAL CORPORATION (JP) 2024-02-29 US claimed
EP-4265629-A1 METHOD FOR PRODUCING LIPID PEPTIDE Nissan Chemical Corporation (JP) 2023-10-25 EP claimed
CN-116648455-A Method for preparing lipid peptide 日产化学株式会社 2023-08-25 CN claimed
CN-116615435-A Method for preparing lipid peptide 日产化学株式会社 2023-08-18 CN claimed
EP-2476691-B1 METHOD FOR MANUFACTURING A LIPIDIC PEPTIDE COMPOUND NISSAN CHEMICAL IND LTD (JP) 2018-01-03 EP claimed
US-9180201-B2 Method for preparing lipopeptide compound NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2015-11-10 US claimed
US-20120253012-A1 METHOD FOR PREPARING LIPOPEPTIDE COMPOUND NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2012-10-04 US claimed
EP-2476691-A1 METHOD FOR MANUFACTURING A LIPIDIC PEPTIDE COMPOUND Nissan Chemical Industries, Ltd. (JP) 2012-07-18 EP claimed
US-20110183913-A1 NOVEL LIPID DIPEPTIDE AND GEL NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-07-28 US claimed
EP-2319894-A1 NOVEL LIPID DIPEPTIDE AND GEL Nissan Chemical Industries, Ltd. (JP) 2011-05-11 EP claimed
US-20240116979-A1 METHOD FOR PRODUCING LIPIDIC PEPTIDE NISSAN CHEMICAL CORPORATION (JP) 2024-04-11 US disclosed
US-20240067675-A1 METHOD FOR PRODUCING LIPID PEPTIDE NISSAN CHEMICAL CORPORATION (JP) 2024-02-29 US disclosed
US-20230404888-A1 COMPOSITION CONTAINING LIPID PEPTIDE AND SUCROSE ESTER NISSAN CHEMICAL CORPORATION (JP) 2023-12-21 US disclosed
EP-4265629-A1 METHOD FOR PRODUCING LIPID PEPTIDE Nissan Chemical Corporation (JP) 2023-10-25 EP disclosed
US-4665066-A BACTERICIDES ELI LILLY AND COMPANY (US) 1987-05-12 US disclosed
EP-0215435-A1 2-Oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-03-25 EP disclosed
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed