SCHEMBL3714654

SCHEMBL3714654

N/C(=N/O)c1ccc(COCC(=O)O)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.41
HDAC2 Q92769 5/20 0.41
RAB9A P51151 4/20 0.41
GAA P10253 3/20 0.41
ALDH1A1 P00352 2/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
PARP10 Q53GL7 2/20 0.40
KDM1A O60341 1/20 0.40
NPC1 O15118 3/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
GFER P55789 1/20 0.40
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714657 1.00 HDAC1 (0.41) HDAC1HDAC2RAB9AGAAALDH1A1
SCHEMBL408726 0.82 KDM1A (0.43) RAB9AALDH1A1KDM1ATP53
SCHEMBL408725 0.82 KDM1A (0.43) RAB9AALDH1A1KDM1ATP53
SCHEMBL10249347 0.80 RAB9A (0.38) HDAC1HDAC2RAB9AGAAALDH1A1
SCHEMBL28860807 0.79 ALDH1A1 (0.61) RAB9AALDH1A1NPC1POLBTP53
SCHEMBL20597672 0.78 KMT2A (0.46) HDAC1HDAC2RAB9AGAAPARP10
SCHEMBL20597670 0.78 KMT2A (0.46) HDAC1HDAC2RAB9AGAAPARP10
SCHEMBL28572177 0.78 KMT2A (0.46) HDAC1HDAC2RAB9AGAAPARP10
SCHEMBL20597699 0.78 HDAC1 (0.45) HDAC1HDAC2RAB9AGAAALDH1A1
SCHEMBL20597701 0.78 HDAC1 (0.45) HDAC1HDAC2RAB9AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414341-B1 OXADIAZOLE DERIVATIVES MERCK SERONO SA (CH) 2017-09-13 EP disclosed
EP-2414342-B1 OXADIAZOLE DERIVATIVES MERCK SERONO SA (CH) 2017-05-31 EP disclosed
US-8815919-B2 Oxadiazole derivatives MERCK SERONO SA (CH) 2014-08-26 US disclosed
US-8802704-B2 Oxadiazole derivatives MERCK SERONO SA (CH) 2014-08-12 US disclosed
WO-2010115751-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed