SCHEMBL3714865

SCHEMBL3714865

CCc1cc(C#N)cc(CC)c1OCC(O)CN

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
ALOX15 P16050 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
KCNH2 Q12809 2/20 0.33
ABCB11 O95342 1/20 0.33
NR2E1 Q9Y466 1/20 0.33
CHEK1 O14757 1/20 0.32
PGR P06401 1/20 0.32
KCNJ5 P48544 1/20 0.32
KCNJ3 P48549 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714866 1.00 TSHR (0.47) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL1175396 0.92 TSHR (0.49) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL1175393 0.92 TSHR (0.49) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL773113 0.82 TSHR (0.60) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL1176040 0.72 S1PR1 (0.54)
SCHEMBL1176038 0.72 S1PR1 (0.54)
SCHEMBL5965751 0.71 ALDH1A1 (0.59) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL5965750 0.71 ALDH1A1 (0.59) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL772719 0.71 ALDH1A1 (0.59) TSHRALOX15SMN1; SMN2KMT2AALDH1A1
SCHEMBL28040009 0.70 PGR (0.32) ALDH1A1KCNH2PGRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222667-A2 NOVEL THIOPHENE DERIVATIVES AS AGONISTS OF S1P1/EDG1 Actelion Pharmaceuticals Ltd. (CH) 2010-09-01 EP disclosed
WO-2009074950-A2 THIOPHENE DERIVATIVES AS AGONISTS OF S1P1/EDG1 ACTELION PHARMACEUTICALS LTD (CH) 2009-06-18 WO disclosed