SCHEMBL3715690

SCHEMBL3715690

O=Cc1ccc2c(c1)CN(C(=O)O)CCO2

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.44
GPR142 Q7Z601 6/20 0.43
PIK3CA P42336 3/20 0.43
CREBBP Q92793 6/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3761090 0.81 RIPK1 (0.47) RIPK1PIK3CACREBBP
SCHEMBL3789225 0.80 RIPK1 (0.46) RIPK1GPR142PIK3CACREBBPCYP2D6
SCHEMBL7968822 0.77 ESR1 (0.44) ALDH1A1KDM4E
SCHEMBL16634768 0.77 ESR2 (0.44) ALDH1A1
SCHEMBL29501124 0.76 RIPK1 (0.54) RIPK1GPR142PIK3CAALDH1A1KDM4E
SCHEMBL17957763 0.76 RIPK1 (0.54) RIPK1GPR142PIK3CAALDH1A1KDM4E
SCHEMBL25228696 0.76 HDAC1 (0.43) ALDH1A1KDM4E
SCHEMBL19644437 0.72 CREBBP (0.60) GPR142PIK3CACREBBP
SCHEMBL3806238 0.72 ROCK1 (0.45) RIPK1GPR142PIK3CACREBBP
SCHEMBL4012679 0.72 RIPK1 (0.45) RIPK1GPR142PIK3CACREBBPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed