SCHEMBL3715977

SCHEMBL3715977

Nc1nc(Cl)cc(CCc2ccccc2)n1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 3/20 0.56
HSP90AA1 P07900 2/20 0.54
KDM4E B2RXH2 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.51
BACE1 P56817 2/20 0.50
DHFR P00374 1/20 0.49
KCNH2 Q12809 1/20 0.48
ADCY10 Q96PN6 6/20 0.48
NOS1 P29475 1/20 0.47
HRH4 Q9H3N8 1/20 0.46
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718901 0.86 HSP90AB1 (0.74) HSP90AB1HSP90AA1KDM4ESMN1; SMN2ADCY10
SCHEMBL28845377 0.82 NOS1 (0.53) BACE1DHFRKCNH2NOS1CYP2D6
SCHEMBL5674666 0.82 KCNH2 (0.52) SMN1; SMN2BACE1KCNH2NOS1
SCHEMBL30509728 0.79 BACE1 (0.51) KDM4EBACE1DHFRKCNH2NOS1
SCHEMBL13153731 0.79 NOS1 (0.51) KDM4EBACE1DHFRKCNH2NOS1
SCHEMBL1998718 0.79 HSP90AB1 (0.51) HSP90AB1HSP90AA1KDM4ESMN1; SMN2DHFR
SCHEMBL28335587 0.76 SMN1; SMN2 (0.63) HSP90AB1HSP90AA1KDM4ESMN1; SMN2DHFR
SCHEMBL4639838 0.75 PRMT6 (0.45) HSP90AB1HSP90AA1KDM4EBACE1
SCHEMBL12122637 0.74 SMN1; SMN2 (0.74) HSP90AB1HSP90AA1KDM4ESMN1; SMN2HRH4
SCHEMBL5745860 0.74 HSP90AB1 (0.53) HSP90AB1HSP90AA1KDM4ESMN1; SMN2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120854-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-10-21 WO disclosed
WO-2010120854-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-10-21 WO disclosed