SCHEMBL3716447

SCHEMBL3716447

CN(Cc1ccccc1)c1cc(C(=O)NO)cc(-c2ccc(C#Cc3cccnc3)cc2)n1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 8/20 0.50
HDAC1 Q13547 7/20 0.47
PTGES O14684 3/20 0.45
AKR1C3 P42330 2/20 0.41
FFAR1 O14842 1/20 0.41
HIF1A Q16665 2/20 0.40
EPAS1 Q99814 2/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
TP53 P04637 1/20 0.39
ACACB O00763 1/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3715131 0.89 HDAC6 (0.46) HDAC6HDAC1PTGESAKR1C3FFAR1
SCHEMBL3721790 0.87 HDAC6 (0.41) HDAC6HDAC1PTGESAKR1C3FFAR1
SCHEMBL13188231 0.86 CSF1R (0.38) HDAC6HDAC1PTGESAKR1C3FFAR1
SCHEMBL3714462 0.84 HDAC6 (0.39) HDAC6HDAC1PTGESAKR1C3FFAR1
Trifluoroacetic Acid SCHEMBL3719131 0.83 FFAR1 (0.39) HDAC6HDAC1PTGESAKR1C3FFAR1
SCHEMBL3719846 0.82 CSF1R (0.40) HDAC6PTGESAKR1C3FFAR1ACACB
SCHEMBL3710041 0.81 HDAC1 (0.46) HDAC6HDAC1PTGESFFAR1HIF1A
SCHEMBL13188474 0.79 CAMK2D (0.47) HDAC6HDAC1FFAR1HIF1AEPAS1
SCHEMBL3716099 0.79 FFAR1 (0.41) HDAC6HDAC1PTGESFFAR1HIF1A
SCHEMBL3716452 0.78 FFAR1 (0.40) PTGESFFAR1HIF1AEPAS1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed