SCHEMBL3716644

SCHEMBL3716644

[CH2]CCc1cccc(F)c1C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.39
AOC3 Q16853 1/20 0.36
P2RX7 Q99572 1/20 0.35
ACHE P22303 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
IDO1 P14902 2/20 0.32
SGMS2 Q8NHU3 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
MEN1 O00255 1/20 0.32
EPHX2 P34913 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
SCN8A Q9UQD0 1/20 0.31
RIPK1 Q13546 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5705869 0.81 TAAR1 (0.61) TAAR1AOC3SMN1; SMN2CD274MAPT
SCHEMBL8097092 0.81 ALDH1A1 (0.42) TAAR1AOC3P2RX7ACHEALDH1A1
Ammonia Solution, Strong SCHEMBL6195329 0.79 ALDH1A1 (0.41) TAAR1AOC3P2RX7ACHEALDH1A1
SCHEMBL27869414 0.79 TAAR1 (0.39) TAAR1AOC3P2RX7ACHEALDH1A1
Hydrochloric Acid SCHEMBL14157235 0.79 TAAR1 (0.59) TAAR1AOC3SMN1; SMN2IDO1CD274
SCHEMBL5584389 0.78 TAAR1 (0.41) TAAR1AOC3GAAIDO1LMNA
SCHEMBL1610124 0.78 ESR1 (0.42) TAAR1P2RX7ACHEALDH1A1GAA
SCHEMBL840509 0.78 TAAR1 (0.62) TAAR1AOC3ALDH1A1IDO1LMNA
SCHEMBL8090805 0.78 TYR (0.40) TAAR1ALDH1A1GAA
SCHEMBL6195324 0.78 MPO (0.49) TAAR1AOC3IDO1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010131146-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO claimed
WO-2010131145-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO claimed
WO-2010131147-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO claimed
WO-2010131145-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed
WO-2010131147-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed