SCHEMBL3716705

SCHEMBL3716705

O=C(NO)c1cncc(-c2ccc(OCc3ccccc3)cc2)c1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 9/20 0.62
HDAC1 Q13547 5/20 0.56
KDM1A O60341 2/20 0.56
SCN2A Q99250 1/20 0.54
SCN10A Q9Y5Y9 1/20 0.54
RAB9A P51151 1/20 0.53
KAT6A Q92794 1/20 0.50
HDAC3 O15379 1/20 0.50
APP P05067 1/20 0.50
ACHE P22303 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
SIRT2 Q8IXJ6 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3711921 0.85 CYP11B1 (0.57) SMPD1SCN2ASCN10ARAB9ASIRT2
SCHEMBL3711432 0.83 HDAC8 (0.56) SMPD1HDAC1KDM1ASCN2ASCN10A
SCHEMBL13187778 0.81 HDAC8 (0.64) HDAC1KDM1ASCN2ASCN10AKAT6A
SCHEMBL443547 0.79 NPC1 (0.65) HDAC1KDM1ASCN2ASCN10ARAB9A
SCHEMBL5944125 0.79 SMPD1 (0.79) SMPD1HDAC1HDAC4HDAC8HDAC6
SCHEMBL3713068 0.78 HDAC1 (0.82) SMPD1HDAC1KDM1ARAB9AKAT6A
SCHEMBL31418277 0.78 ALDH1A1 (0.51) SMPD1SCN2ASCN10ARAB9ASIRT2
SCHEMBL3715274 0.78 SMPD1 (0.67) SMPD1HDAC1
SCHEMBL10839211 0.77 SMPD1 (0.74) SMPD1HDAC1HDAC3APPACHE
SCHEMBL1608032 0.76 SMPD1 (1.00) SMPD1HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed