SCHEMBL3717840

SCHEMBL3717840

NCCC(N)c1ccncn1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
P2RX7 Q99572 1/20 0.35
LOXL2 Q9Y4K0 3/20 0.34
CYP19A1 P11511 1/20 0.33
DPP4 P27487 1/20 0.32
HRH1 P35367 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26695870 0.85 HSP90AA1 (0.38) HSP90AA1P2RX7CYP19A1
SCHEMBL11813334 0.82 CYP2D6 (0.41) HSP90AA1P2RX7CYP19A1
SCHEMBL2894352 0.80 HSP90AA1 (0.40) HSP90AA1P2RX7CYP19A1
SCHEMBL5669611 0.80 P2RX7 (0.43) HSP90AA1P2RX7CYP19A1
Ammonia Solution, Strong SCHEMBL3717839 0.78 HSP90AA1 (0.39) HSP90AA1P2RX7CYP19A1
SCHEMBL28804110 0.77 HSP90AA1 (0.32) HSP90AA1
SCHEMBL16150460 0.74 P2RX7 (0.42) HSP90AA1P2RX7CYP19A1
SCHEMBL3224199 0.73 HRH1 (0.45) HRH1
SCHEMBL3718708 0.72
SCHEMBL28864538 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010131147-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed
WO-2010131145-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed
WO-2010131146-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed