SCHEMBL3718197

SCHEMBL3718197

NC(=O)c1ccc(-c2cn[nH]c2)cc1OCCN1CCCC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.57
ROCK1 Q13464 3/20 0.57
CDC42BPA Q5VT25 1/20 0.51
MELK Q14680 1/20 0.49
PARP1 P09874 2/20 0.46
DHODH Q02127 1/20 0.46
CHEK1 O14757 1/20 0.46
MKNK1 Q9BUB5 3/20 0.46
MKNK2 Q9HBH9 3/20 0.46
CHEK2 O96017 1/20 0.45
HTR3A P46098 1/20 0.42
DRD2 P14416 1/20 0.41
DRD1 P21728 1/20 0.41
DRD3 P35462 1/20 0.41
HTR1A P08908 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718200 0.83 ROCK2 (0.61) ROCK2ROCK1CDC42BPAHTR3A
SCHEMBL3807004 0.82 ROCK2 (0.43) ROCK2ROCK1CDC42BPAMELKPARP1
SCHEMBL3801724 0.79 HTT (0.54) ROCK2ROCK1MELKMKNK1MKNK2
SCHEMBL3713988 0.79 ROCK2 (0.69) ROCK2ROCK1CDC42BPAMELK
SCHEMBL20290838 0.77 MELK (0.70) ROCK2ROCK1CDC42BPAMELKMKNK2
SCHEMBL3243986 0.76 ROCK2 (0.66) ROCK2ROCK1CDC42BPAMELK
SCHEMBL3714539 0.75 MELK (0.56) ROCK2ROCK1MELKMKNK1MKNK2
SCHEMBL3722812 0.75 MELK (0.55) ROCK2ROCK1MELKPARP1MKNK1
SCHEMBL3656437 0.75 MKNK2 (0.61) ROCK2ROCK1MELKMKNK1MKNK2
SCHEMBL13885328 0.75 PSMB1 (0.54) CHEK1CHEK2DRD2DRD1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed