SCHEMBL3718255

SCHEMBL3718255

COc1ccc(Oc2ccc(N(C)C(=O)C3(NC(=O)c4cncc(C)c4)CC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
RAF1 P04049 3/20 0.34
BDKRB1 P46663 1/20 0.33
GPBAR1 Q8TDU6 2/20 0.33
EPHX2 P34913 3/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
MITF O75030 1/20 0.32
TP53 P04637 1/20 0.32
RAB9A P51151 1/20 0.32
FAAH O00519 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
SSTR5 P35346 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3728515 0.92 EPHX2 (0.35) GAAMAPTRAF1BDKRB1EPHX2
SCHEMBL3722520 0.92 BDKRB1 (0.41) GAAMAPTMAPK1RAF1BDKRB1
SCHEMBL3722273 0.92 PPARG (0.35) GAARAF1BDKRB1EPHX2
SCHEMBL3729297 0.85 KMT2A (0.35) GAAMAPTMAPK1EPHX2KDM4E
SCHEMBL3795493 0.85 GAA (0.34) GAAGPBAR1FAAHPROKR1
SCHEMBL13191233 0.84 BDKRB1 (0.44) BDKRB1EPHX2
SCHEMBL3722724 0.84 MEN1 (0.36) GAARAF1BDKRB1GPBAR1EPHX2
SCHEMBL3718253 0.83 GAA (0.33) GAAMAPTEPHX2KDM4EPROKR1
SCHEMBL3719005 0.83 MAPK10 (0.35) GAAMAPTKDM4E
SCHEMBL3801380 0.82 CNR1 (0.42) BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed