SCHEMBL3728515

SCHEMBL3728515

COc1ccc(Oc2ccc(N(C)C(=O)C3(NC(=O)c4cncc(F)c4)CC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.35
ABL1 P00519 2/20 0.34
CNR1 P21554 1/20 0.34
RAF1 P04049 3/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
BDKRB1 P46663 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GAA P10253 1/20 0.33
MAPK10 P53779 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722520 0.92 BDKRB1 (0.41) EPHX2RAF1KDM4EMAPTBDKRB1
SCHEMBL3718255 0.92 GAA (0.34) EPHX2RAF1KDM4EMAPTBDKRB1
SCHEMBL3722273 0.92 PPARG (0.35) EPHX2CNR1RAF1BDKRB1GAA
SCHEMBL3795493 0.85 GAA (0.34) CYP1A2CYP3A4GAAMAPK10PROKR1
SCHEMBL3728513 0.84 BDKRB1 (0.44) EPHX2ABL1CNR1BDKRB1
SCHEMBL3718253 0.83 GAA (0.33) EPHX2KDM4EMAPTCYP1A2GAA
SCHEMBL3729297 0.83 KMT2A (0.35) EPHX2CNR1KDM4EMAPTGAA
SCHEMBL3719005 0.83 MAPK10 (0.35) KDM4EMAPTGAAMAPK10
SCHEMBL3722724 0.82 MEN1 (0.36) EPHX2CNR1RAF1BDKRB1L3MBTL1
SCHEMBL3718996 0.82 CNR1 (0.44) CNR1BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed