SCHEMBL3718310

SCHEMBL3718310

CN(C)c1c(-c2ccc(C#Cc3cccnc3)cc2)cc2ccncc2c1C(=O)NO

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 1/20 0.39
FFAR1 O14842 1/20 0.37
PTGES O14684 3/20 0.36
AKR1C3 P42330 2/20 0.36
XIAP P98170 3/20 0.36
BIRC2 Q13490 3/20 0.36
GRM5 P41594 2/20 0.36
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CYP2A6 P11509 1/20 0.34
MAPT P10636 1/20 0.34
SNCA P37840 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3713867 0.89 ALDH2 (0.38) ALDH2FFAR1PTGESAKR1C3XIAP
SCHEMBL3721286 0.85 FFAR1 (0.39) ALDH2FFAR1XIAPBIRC2GRM5
SCHEMBL3714355 0.80 MMP2 (0.42) HDAC1HDAC6
SCHEMBL13188252 0.77 FFAR1 (0.41) FFAR1PTGESXIAPBIRC2GRM5
SCHEMBL3721229 0.77 SLC2A1 (0.39) ALDH2FFAR1XIAPBIRC2GRM5
SCHEMBL3721790 0.73 HDAC6 (0.41) FFAR1PTGESAKR1C3GRM5CHRNB2
SCHEMBL3715059 0.72 SLC2A1 (0.39) ALDH2FFAR1PTGESAKR1C3XIAP
SCHEMBL3716448 0.71 TNIK (0.42) FFAR1PTGESAKR1C3GRM5CHRNB2
SCHEMBL3713900 0.71 GRM5 (0.40) ALDH2FFAR1GRM5CYP2A6
SCHEMBL3721418 0.71 CCNC (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed