SCHEMBL3718608

SCHEMBL3718608

O=Cc1occc1-c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.46
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
PTGS1 P23219 4/20 0.40
PTGS2 P35354 7/20 0.37
TDO2 P48775 1/20 0.34
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NR4A2 P43354 1/20 0.33
NOTUM Q6P988 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8172271 0.81 PTGS2 (0.33) KDM4EALDH1A1PTGS2NPC1RAB9A
SCHEMBL9586893 0.81 CYP2A6 (0.40) KDM4EALDH1A1LMNAPTGS1PTGS2
SCHEMBL3132305 0.80 MEN1 (0.37) ALDH1A1RAB9AMEN1KMT2AHPGD
SCHEMBL27431758 0.77 HRH3 (0.43)
SCHEMBL27933553 0.75 APP (0.44) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL30541683 0.74 APP (0.43) KDM4EALDH1A1MEN1KMT2A
SCHEMBL31571399 0.73 NPC1 (0.34) ALDH1A1NPC1SMN1; SMN2
SCHEMBL5132966 0.72 NOTUM (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL10950612 0.71 MAPK14 (0.79) MAPK14KDM4EALDH1A1PTGS1PTGS2
SCHEMBL14398163 0.71 KEAP1 (0.39) KDM4EALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129848-A2 2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXAMIDES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-11 WO disclosed
WO-2008005651-A2 CYCLIC CARBOXYLIC ACID RHODANINE DERIVATIVES FOR THE TREATMENT AND PREVENTION OF TUBERCULOSIS DECODE CHEMISTRY, INC. (US) 2008-01-10 WO disclosed