SCHEMBL3718709

SCHEMBL3718709

NCc1occc1-c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.46
LOXL2 Q9Y4K0 3/20 0.40
HTR2C P28335 1/20 0.38
TDO2 P48775 1/20 0.38
MAOB P27338 1/20 0.37
PTGS1 P23219 3/20 0.33
PTGS2 P35354 3/20 0.33
TAAR1 Q96RJ0 3/20 0.33
NOTUM Q6P988 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAOA P21397 2/20 0.32
LOX P28300 1/20 0.32
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
ADORA2A P29274 1/20 0.31
PIK3R1 P27986 1/20 0.31
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4652501 0.80 DPP4 (0.47) LOXL2TDO2TAAR1NOTUMRAB9A
SCHEMBL10950612 0.71 MAPK14 (0.79) MAPK14TDO2PTGS1PTGS2NOTUM
SCHEMBL16807848 0.69 MAPK14 (0.50) MAPK14TDO2PTGS2NOTUMNPC1
SCHEMBL3718608 0.69 MAPK14 (0.46) MAPK14TDO2PTGS1PTGS2NOTUM
SCHEMBL6633897 0.68 MAPK14 (0.45) MAPK14TDO2PTGS1NPC1RAB9A
SCHEMBL8138770 0.65 BCL2L1 (0.48) MAPK14NPC1RAB9A
SCHEMBL3761020 0.64 LOXL2 (0.43) LOXL2HTR2CTDO2MAOBPTGS1
SCHEMBL3723618 0.64 DPP4 (0.69) MAPK14LOXL2HTR2CMAOBPTGS1
SCHEMBL8133757 0.63 MAPK14 (1.00) MAPK14
SCHEMBL7457056 0.63 LOXL2 (0.30) LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129848-A2 2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXAMIDES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-11 WO disclosed