SCHEMBL3719583

SCHEMBL3719583

CC(=O)NC(C)(I)c1ccc2cc(Oc3ccc(OCC(F)(F)F)cc3C)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
PPARD Q03181 9/20 0.41
CYP2C9 P11712 2/20 0.40
CYP1A2 P05177 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP17A1 P05093 2/20 0.38
CYP2C19 P33261 1/20 0.38
PPARA Q07869 3/20 0.37
FFAR1 O14842 1/20 0.37
POLB P06746 1/20 0.37
PPARG P37231 2/20 0.37
RAB9A P51151 1/20 0.37
SSTR4 P31391 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724597 0.84 PPARA (0.41) ALDH1A1PPARDCYP2C9CYP1A2KDM4E
SCHEMBL3722840 0.79 MEN1 (0.45) ALDH1A1CYP2C9CYP1A2KDM4ERAB9A
SCHEMBL3721105 0.77 THRB (0.34) ALDH1A1PPARDPPARAPPARG
SCHEMBL3726321 0.77 CYP2C9 (0.52) ALDH1A1CYP2C9CYP1A2KDM4ECYP17A1
SCHEMBL3726323 0.77 SMN1; SMN2 (0.43) ALDH1A1CYP2C9CYP1A2KDM4EPOLB
SCHEMBL3727217 0.76 MEN1 (0.38) ALDH1A1CYP2C9CYP1A2KDM4ECYP2C19
SCHEMBL3717756 0.76 SCN9A (0.41) ALDH1A1CYP2C9CYP1A2KDM4ECYP2C19
SCHEMBL3725363 0.74 ESRRA (0.47) FFAR1PPARG
SCHEMBL3719849 0.73 KDM4E (0.44) CYP1A2KDM4ERAB9A
SCHEMBL3720547 0.72 SCN7A (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed