SCHEMBL3720294

SCHEMBL3720294

CC(=O)NC(C)c1ccc2cc(Oc3ccc(OCC(F)(F)F)cc3Cl)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 17/20 0.43
CACNA1G O43497 1/20 0.42
CACNA1H O95180 1/20 0.42
CNR2 P34972 1/20 0.42
KCNH2 Q12809 1/20 0.42
CACNA1I Q9P0X4 1/20 0.42
ACACA Q13085 4/20 0.41
CYP2C9 P11712 5/20 0.40
CYP3A4 P08684 2/20 0.40
SCN9A Q15858 1/20 0.40
CYP2C19 P33261 2/20 0.40
CYP17A1 P05093 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718634 0.86 CYP17A1 (0.51) ACACBCACNA1GCACNA1HCNR2KCNH2
SCHEMBL3726420 0.86 ACACB (0.47) ACACBKCNH2ACACA
SCHEMBL3728856 0.84 ACACB (0.42) ACACBACACA
SCHEMBL3720296 0.81 SCN9A (0.45) CYP2C9SCN9A
SCHEMBL3717756 0.79 SCN9A (0.41) CYP2C9CYP3A4SCN9ACYP2C19
SCHEMBL3720848 0.79 CYP17A1 (0.46) ACACBACACACYP2C9CYP2C19CYP17A1
SCHEMBL3727616 0.76 ESRRA (0.52) CYP2C9CYP2C19CYP17A1
SCHEMBL3726321 0.75 CYP2C9 (0.52) ACACBACACACYP2C9CYP2C19CYP17A1
SCHEMBL3718635 0.74 PPARA (0.45) ACACBCYP2C9SCN9A
SCHEMBL13077221 0.74 ACACB (0.57) ACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO claimed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed