SCHEMBL3726420

SCHEMBL3726420

COc1ccc(Oc2ccc3nc(C(C)NC(C)=O)ccc3c2)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 10/20 0.47
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
HTR2A P28223 1/20 0.40
SLC6A4 P31645 1/20 0.40
KCNH2 Q12809 1/20 0.40
HPGDS O60760 2/20 0.40
ACACA Q13085 1/20 0.40
CHEK2 O96017 1/20 0.39
PNLIP P16233 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3728856 0.90 ACACB (0.42) ACACBACACA
SCHEMBL3720294 0.86 ACACB (0.43) ACACBKCNH2ACACA
SCHEMBL3798078 0.84 ALOX5 (0.57) ACACBTAS1R3TAS1R1ACACA
SCHEMBL3717394 0.79 HDAC8 (0.44) KCNH2CHEK2PNLIPHDAC3HDAC4
SCHEMBL3726423 0.77 MTNR1A (0.47)
SCHEMBL3722350 0.76 TAS1R3 (0.56) ACACBTAS1R3TAS1R1ACACA
SCHEMBL3721369 0.75 ALDH1A1 (0.50) ACACBACACA
SCHEMBL3719663 0.75 ACACB (0.56) ACACBTAS1R3TAS1R1ACACA
SCHEMBL3724748 0.74 ACACB (0.47) ACACBACACA
SCHEMBL3726987 0.73 ACACB (0.48) ACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed